All Pages : 675 ; Current Page : 13 ; Activities from 121 to 130
NR Protein | Protein Name | Ligand ID | Ligand Name | EC 50 |
---|---|---|---|---|
NR1C1 | Peroxisome proliferator activated receptor alpha | 7645 | (2S)-2-[(4-{3-[2-chloro-4-(2,2,2-trifluoroethoxy)phenoxy]propoxy}phenyl)methyl]-2-methylbutanoic acid | 0.008 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 8994 | 5-({3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl}methyl)-1-(propoxycarbonyl)-1,2,3,4-tetrahydropyridine-4-carboxylic acid | 0.008 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 9004 | (2S,3S)-1-(4-tert-butylphenyl)-3-[(3-{2-[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]ethoxy}phenyl)methyl]-4-oxoazetidine-2-carboxylic acid | 0.008 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 10843 | 2-[4-[2-[cyclohexylcarbamoyl-[2-(4-phenylphenyl)ethyl]amino]ethyl]phenyl]sulfanyl-2-methylpropanoic acid | 0.008 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 11136 | 2-{4-[({[2-(3-bromophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(furan-2-ylmethyl)amino)methyl]phenoxy}-2-methylpropanoic acid | 0.008 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 11290 | 5-({3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl}methyl)-1-[(2-methylpropoxy)carbonyl]-1,2,3,4-tetrahydropyridine-4-carboxylic acid | 0.009 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 11237 | 2-{[(3-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methoxy}phenyl)methyl](4-methylphenoxycarbonyl)amino}acetic acid | 0.009 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 11325 | 2-{[(3-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)methyl][(cyclopentyloxy)carbonyl]amino}acetic acid | 0.009 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 11248 | 2-({[3-({5-methyl-2-[4-(propan-2-yl)phenyl]-1,3-oxazol-4-yl}methoxy)phenyl]methyl}(4-methylphenoxycarbonyl)amino)acetic acid | 0.009 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 7598 | (2S)-2-methyl-3-(4-{2-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]ethoxy}phenyl)-2-phenoxypropanoic acid | 0.009 |
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