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NR Protein | Protein Name | Ligand ID | Ligand Name | EC 50 |
---|---|---|---|---|
NR1C1 | Peroxisome proliferator activated receptor alpha | 9176 | (2S)-2-({4-[3-(2-chloro-4-cyclohexylphenoxy)propoxy]phenyl}methyl)-2-methylbutanoic acid | 0.001 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 9215 | (2s,5s)-2-methyl-5-[(4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}phenyl)methyl]-1,3-dioxane-2-carboxylic acid | 0.001 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 9265 | (4Z)-4-[({6-[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]hexyl}oxy)imino]-4-phenylbutanoic acid | 0.001 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 9349 | (2s,5s)-2-methyl-5-({4-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methoxy]phenyl}methyl)-1,3-dioxane-2-carboxylic acid | 0.001 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 10840 | 2-[4-[2-[4-cyclohexylbutyl-[(3,5-dichlorophenyl)carbamoyl]amino]ethyl]phenyl]sulfanyl-2-methylpropanoic acid | 0.001 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 10890 | 5-[(4-ethoxy-3-methylphenyl)sulfanylmethyl]-4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole | 0.001 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 3549 | 2-(4-{3-[(3-phenyl-7-propyl-1,2-benzoxazol-6-yl)oxy]propoxy}phenoxy)propanoic acid | 0.002 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 3653 | 2-(4-{3-[(3-phenyl-7-propyl-1,2-benzoxazol-6-yl)oxy]propoxy}-1H-indol-1-yl)acetic acid | 0.002 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 3915 | (2S)-3-(4-{[(2E)-3-[3,5-bis(2,2,2-trifluoroethoxy)phenyl]prop-2-en-1-yl]oxy}phenyl)-2-ethoxypropanoic acid | 0.002 |
NR1C1 | Peroxisome proliferator activated receptor alpha | 3945 | 2-methyl-2-(4-{4-[(3-phenyl-7-propyl-1,2-benzoxazol-6-yl)oxy]butoxy}phenoxy)propanoic acid | 0.002 |
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