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NR Protein | Protein Name | Ligand ID | Ligand Name | EC 50 |
---|---|---|---|---|
NR2B1 | Retinoid X receptor alpha | 3298 | (E)-3-[3-[2-ethoxy-3,5-di(propan-2-yl)phenyl]thieno[2,3-c]pyridin-5-yl]but-2-enoic acid | 1.442 |
NR2B1 | Retinoid X receptor alpha | 3301 | (E)-3-[3-[2-butoxy-3,5-di(propan-2-yl)phenyl]-1-methylindol-5-yl]but-2-enoic acid | 1.533 |
NR2B1 | Retinoid X receptor alpha | 6073 | 4-(3-fluoro-5,5,8,8-tetramethyl-6,7-dihydronaphthalene-2-carbonyl)benzoic acid | 1.82 |
NR2B1 | Retinoid X receptor alpha | 6148 | 2-(N-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)methylsulfonamido)pyrimidine-5-carboxylic acid | 1.888 |
NR2B1 | Retinoid X receptor alpha | 3369 | (2E, 4E, 6E)-7-(3,5-Di-trifluoromethylphenyl)-3-methylocta-2,4,6-trienoic acid | 2.007 |
NR2B1 | Retinoid X receptor alpha | 6077 | 4-(3-methoxy-5,5,8,8-tetramethyl-6,7-dihydronaphthalene-2-carbonyl)benzoic acid | 2.019 |
NR2B1 | Retinoid X receptor alpha | 6145 | 4-(N-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)propylsulfonamido)benzoic acid | 2.019 |
NR2B1 | Retinoid X receptor alpha | 3455 | 5-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalene-2-carbonyl)thiophene-2-carboxylic acid | 2.2 |
NR2B1 | Retinoid X receptor alpha | 6061 | 2-[(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)sulfanyl]-1,3-thiazole-5-carboxylic acid | 2.3 |
NR2B1 | Retinoid X receptor alpha | 5982 | 4-[1-(3,8,8-trimethyl-6,7-dihydro-5H-naphthalen-2-yl)ethenyl]benzoic acid | 2.4 |
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