7300 : 4-methyl-N-[(4-trifluoromethanesulfonamidophenyl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxamide
Ligand Basic Message
| Ligand | Scaffold |
|---|---|
 |  |
| ID | 7300 |
| Name | 4-methyl-N-[(4-trifluoromethanesulfonamidophenyl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxamide |
| smile | CC1N=C(C2=CC=C(C(F)(F)F)C=C2)SC=1C(NCC1=CC=C(C=C1)NS(C(F)(F)F)(=O)=O)=O |
| weight | 523 |
| scaffold ID | 174 |
| scaffold smile | O=C(NCc1ccccc1)c1cnc(-c2ccccc2)s1 |
Ligand Activities
| NR Protein | Protein Name | Ligand ID | Ligand Name | EC 50 |
|---|---|---|---|---|
| NR1C3 | Peroxisome proliferator activated receptor gamma | 7300 | 4-methyl-N-[(4-trifluoromethanesulfonamidophenyl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxamide | 0.5 |
Scaffold Activities Statistic