Target Description

Type Detail
Target ID T23RWU
Protein Name Type-1 angiotensin II receptor
Uniprot ID P30556
Protein Name Alias AT1AR;  AT1BR;  Angiotensin II type-1 receptor;  AT1
Gene ID 185
Gene Symbol AGTR1
Gene Alias AGTR1A;  AGTR1B;  AT2R1;  AT2R1B
TTD T74456: Successful target
Pfam PF00001
GO
0007200:phospholipase C-activating G protein-coupled receptor signaling pathway

0042127:regulation of cell population proliferation

0002018:renin-angiotensin regulation of aldosterone production

0016021:integral component of membrane

1903589:positive regulation of blood vessel endothelial cell proliferation involved in sprouting angiogenesis

0038166:angiotensin-activated signaling pathway

0033864:positive regulation of NAD(P)H oxidase activity

0050727:regulation of inflammatory response

0050729:positive regulation of inflammatory response

0004945:angiotensin type II receptor activity

0006954:inflammatory response

0086097:phospholipase C-activating angiotensin-activated signaling pathway

0007204:positive regulation of cytosolic calcium ion concentration

0046982:protein heterodimerization activity

0019229:regulation of vasoconstriction

0051482:positive regulation of cytosolic calcium ion concentration involved in phospholipase C-activating G protein-coupled signaling pathway

0019722:calcium-mediated signaling

0010873:positive regulation of cholesterol esterification

0034374:low-density lipoprotein particle remodeling

0060326:cell chemotaxis

0002034:maintenance of blood vessel diameter homeostasis by renin-angiotensin

0001558:regulation of cell growth

0003081:regulation of systemic arterial blood pressure by renin-angiotensin

0010744:positive regulation of macrophage derived foam cell differentiation

0035813:regulation of renal sodium excretion

0004930:G protein-coupled receptor activity

2000379:positive regulation of reactive oxygen species metabolic process

0007266:Rho protein signal transduction

0005886:plasma membrane

0007186:G protein-coupled receptor signaling pathway

0001596:angiotensin type I receptor activity

0005887:integral component of plasma membrane

0031711:bradykinin receptor binding

0097746:blood vessel diameter maintenance

0032430:positive regulation of phospholipase A2 activity

0001822:kidney development

0032270:positive regulation of cellular protein metabolic process

PDB 4YAY ; 6OS1 ; 1ZV0 ; 6DO1 ; 6OS2 ; 6OS0 ; 4ZUD
Drugbank DB01347 ; DB13919 ; DB11842 ; DB01342 ; DB00796 ; DB00966 ; DB09279 ; DB00275 ; DB00678 ; DB01349 ; DB00177 ; DB05739 ; DB00876 ; DB08822 ; DB01029
KEGG hsa:185

Related Compounds  (Total: 8)

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C0055
Name: Estradiol
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C0363
Name: Resveratrol
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C0868
Name: Aldosterone
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C0907
Name: Angiotensin Ii
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C1017
Name: puerarin


Related Herbs  (Total: 71)

Herb idChinese Pin YinChinese CharacterEnglish NameLatin Name
H0437 She Xiang麝香 AbelmuskMoschus moschiferus
H1213 Hu Zhang虎杖 Japanese fleeceflowerPolygonum cuspidatum
H0416 Shan Shen山参 NAPanax ginseng
H0269 Mu Gua木瓜 Chinese floweringquinceChaenomeles sinensis
H0235 Mao She Xiang毛麝香 AbelmuskMoschus moschiferus
H0693 Xue Xie血蝎 Dragon's bloodDaemonorops draco
H1250 Huang Qi Ti Qu Ye黄芪提取液 Membranous milkvetchAstragalus membranaceus
H0111 Ku Shen苦参 Lightyellow sophoraSophora flavescens
H0277 Nan Ban Lan Gen南板蓝根 Indigowoad rootBaphicacanthus cusia
H0236 Mao She Xiang Jin Gao毛麝香浸膏 AbelmuskMoschus moschiferus
H0226 Man Yue Mei蔓越莓 CranberryVaccinium oxycoccos
H0533 Teng Ku Shen藤苦参 NASophora flavescens
H0472 Shu Da Huang熟大黄 NARheum palmatum
H0926 Da Huang大黄 Medicinal rhubarbRheum officinale
H0520 Tai Pan Fen胎盘粉 Fetus powderHuman placenta
H0626 Xi Nan Huang Qin西南黄芩 Yunnan skullcapScutellaria amoena
H0360 Ren Zhong Bai人中白 Human urine sedimentHomo sapiens
H0385 San Qi Ye Jing三七叶茎 SanchiPanax notoginseng
H0883 Chuan She Gan川射干 BlackberrylilyBelamcanda chinensis
H0084 Jiu Li Xiang九里香 Common jasminorangeMurraya paniculata
H0201 Ma Huang Jin Gao麻黄浸膏 Chinese ephedraEphedra sinica
H0927 Da Huang Jin Gao大黄浸膏 Medicinal rhubarbRheum officinale
H0200 Ma Huang Gen麻黄根 Chinese ephedra rootEphedra sinica
H1166 He Shou Wu何首乌 Tuber fleeceflowerPolygonum multiflorum
H0932 Ba Qia菝葜 Chinaroot greenbrierSmilax china
H0356 Ren Gong She Xiang人工麝香 AbelmuskMoschus moschiferus
H0142 Liang Jiang良姜 NAAlpinia officinarum
H0765 Chi Dou赤豆 Assuki beanVigna angularis
H0570 Tu Fu Ling土茯苓 Glabrous greenbrierSmilax glabra
H1247 Huang Qi黄芪 Membranous milkvetchAstragalus membranaceus
H0382 San Qi Hua三七花 SanchiPanax notoginseng
H0434 She Pu Tao蛇葡萄 AmpelopsisAmpelopsis brevipedunculata
H1102 Gu Sui Bu骨碎补 Fortune’s drynaria rhizomeDrynaria fortunei
H0077 Jiu EthanolVinum
H0957 Dang Gui Teng当归藤 NAEmbelia parviflora
H0198 Ma Huang Gao麻黄膏 Chinese ephedraEphedra sinica
H0847 Zi He Che紫河车 Human placentaHomo sapiens
H0928 Da Huang Liu Jin Gao大黄流浸膏 Medicinal rhubarbRheum officinale
H0556 Tie Xian Cao铁线草 NAAdiantum capillus-veneris
H0197 Ma Huang麻黄 Chinese ephedraEphedra sinica
H0270 Mu Hu Die木蝴蝶 Indian trumpetflowerOroxylum indicum
H0521 Tai Pan Zu Zhi Fen胎盘组织粉 NAHuman placenta
H0432 She Gan射干 BlackberrylilyBelamcanda chinensis
H0826 Chu Mu Dan臭牡丹 rose glorybowerClerodendrum bungei
H0153 Ling Zhi(1)灵芝 Lucid ganodermaGanoderma lucidum
H1093 Gao Liang Jiang You高良姜油 Lesser galangalAlpinia officinarum
H0278 Nan Ban Lan Gen Jin Gao Fen南板蓝根浸膏粉 Indigowoad rootBaphicacanthus cusia
H0895 Chuan Yu Jin川郁金 TurmericCurcuma longa
H0661 Xiao Hei Dou小黑豆 Black turtle beanPhaseolus vulgaris
H0358 Ren Shen Ye人参叶 Ginseng leafPanax ginseng
H1117 Guan Zhong贯众 Male fern rhizomeDryopteris crassirhizoma
H0617 Qian Cao Teng茜草藤 NARubia cordifolia
H0383 San Qi Jing Ye三七茎叶 SanchiPanax notoginseng
H0396 Sang Ye桑叶 White mulberry leafMorus alba
H0384 San Qi Ye三七叶 Folium panax notoginsengPanax notoginseng
H0391 Sang Pi桑皮 Prepared root-bark white mulberryMorus alba
H1240 Huang Jing Zi黄荆子 NAVitex negundo
H0761 Yu Jin郁金 AromaticTurmericCurcuma aromatica
H0397 Sang Zhi桑枝 White mulberry branchMorus alba
H0028 Jiang Huang姜黄 Common turmericCurcuma longa
H0357 Ren Shen人参 GinsengPanax ginseng
H0380 San Qi Gan Jin Gao三七干浸膏 SanchiPanax notoginseng
H0555 Tie Xian Cai铁苋菜 Copperleaf herbHerba acalyphae
H1249 Huang Qi Jin Gao黄芪浸膏 Membranous milkvetchAstragalus membranaceus
H0381 San Qi Gao Fen三七膏粉 SanchiPanax notoginseng
H0246 Mi Ma Huang蜜麻黄 Ephedra equisetinEphedra sinica
H1092 Gao Liang Jiang高良姜 Lesser galangalAlpinia officinarum
H0705 Yan Hu Lu Ba盐胡芦巴 FenugreekTrigonella foenum-graecum
H1248 Huang Qi Gan Jin Gao黄芪干浸膏 Membranous milkvetchAstragalus membranaceus
H0575 Tu Ku Shen土苦参 all-grass of hooker wingheadSophora flavescens
H0152 Ling Zhi Jin Gao灵芝浸膏 NAGanoderma lucidum