Target Description

Type Detail
Target ID T36YWU
Protein Name Kelch-like ECH-associated protein 1
Uniprot ID Q14145
Protein Name Alias Cytosolic inhibitor of Nrf2;  INrf2;  Kelch-like protein 19
Gene ID 9817
Gene Symbol KEAP1
Gene Alias INRF2;  KIAA0132;  KLHL19
TTD T83198: Clinical Trial target
Pfam PF01344 ; PF07707 ; PF00651
GO
0008134:transcription factor binding

0042802:identical protein binding

0016567:protein ubiquitination

0097718:disordered domain specific binding

0005829:cytosol

0016234:inclusion body

0034451:centriolar satellite

0034599:cellular response to oxidative stress

0031463:Cul3-RING ubiquitin ligase complex

0005737:cytoplasm

0006511:ubiquitin-dependent protein catabolic process

0005783:endoplasmic reticulum

0030496:midbody

0001701:in utero embryonic development

0045604:regulation of epidermal cell differentiation

0042994:cytoplasmic sequestering of transcription factor

0043433:negative regulation of DNA-binding transcription factor activity

0016032:viral process

0032436:positive regulation of proteasomal ubiquitin-dependent protein catabolic process

0005654:nucleoplasm

0016579:protein deubiquitination

0010506:regulation of autophagy

0071353:cellular response to interleukin-4

0005884:actin filament

0043687:post-translational protein modification

PDB 3VNG ; 6ROG ; 6SP4 ; 4XMB ; 2FLU ; 5WHL ; 5DAF ; 4CXJ ; 5GIT ; 4CXT ; 5WG1 ; 4L7C ; 6W67 ; 5X54 ; 6FMQ ; 6SP1 ; 6W66 ; 5WFV ; 3ZGD ; 5DAD ; 4IFJ ; 6T7Z ; 6Z6A ; 5WHO ; 3VNH ; 4IFL ; 6W69 ; 6LRZ ; 6W68 ; 6FMP ; 4IFN ; 1ZGK ; 6FFM ; 4IQK ; 6WCQ ; 6V6Z ; 6T7V ; 4CXI ; 6UF0 ; 6TYP ; 6HWS ; 5WIY ; 4L7B ; 4N1B ; 5F72 ; 5NLB ; 5WFL ; 4IN4 ; 4L7D ; 1U6D ; 3ZGC ; 6TG8 ; 6TYM
Drugbank DB08908
KEGG hsa:9817

Related Compounds  (Total: 5)

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C0025
Name: Dioscin
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C0045
Name: Epicatechin Gallate
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C0053
Name: Esculetin
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C0058
Name: Ethacrynic Acid
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C0421
Name: Sulforaphane


Related Herbs  (Total: 132)

Herb idChinese Pin YinChinese CharacterEnglish NameLatin Name
H0543 Tian Men Dong天门冬 Cochinchinese asparagusAsparagus cochinchinensis
H1227 Huai Zhi槐枝 NASophora japonica
H1089 Gang Ren Zi岗稔子 rose myrtleRhodomyrtus tomentosa
H0226 Man Yue Mei蔓越莓 CranberryVaccinium oxycoccos
H1015 Du Zhong杜仲 EucommiaEucommia ulmoides
H1128 Bai Jiang败酱 Whiteflower patriniaPatrinia villosa
H0926 Da Huang大黄 Medicinal rhubarbRheum officinale
H0360 Ren Zhong Bai人中白 Human urine sedimentHomo sapiens
H0745 Yin Chen Hao茵陈蒿 Capillary wormwoodArtemisia capillaris
H1034 Fei Yang Cao飞杨草 NAEuphorbia hirta
H1164 He Geng荷梗 Hindu lotus petioleNelumbo nucifera
H0874 Chuan Long Shu Yu穿龙薯蓣 Nippon yamDioscorea nipponica
H0819 Zhi Zi Jin Gao栀子浸膏 Cape jasmine fruitGardenia jasminoides
H0126 Lai Fu Zi莱菔子 Garden radish seedRaphanus sativus
H1114 Guan Gui官桂 CassiabarktreeCinnamomum cassia
H0955 Dang Gui当归 Chinese angelicaAngelica sinensis
H0315 Pu Gong Ying Jin Gao蒲公英浸膏 Mongolian dandelionTaraxacum mongolicum
H0802 Zhi Geng枳梗 NACitrus aurantium
H0551 Cang Zhu苍术 Swordlike atractylodesAtractylodes lancea
H1056 Fu Pen Zi覆盆子 Red-and-Yellow garden raspberryRubus idaeus
H0637 Cha Ye茶叶 Common teaCamellia sinensis
H0804 Zhi Ke枳壳 Seville ora nge unripe fruitCitrus aurantium
H0541 Cang Qie Gen藏茄根 Tibetan eggplant rootAnisodus tanguticus
H0960 Dang Shen Qing Gao党参清膏 Root of hairy asiabellCodonopsis pilosula
H1073 Gan Cao Jie甘草节 Glycyrrhiza uralensis fischGlycyrrhiza uralensis
H0805 Zhi Ke Gan Jin Gao枳壳干浸膏 Seville ora nge unripe fruitCitrus aurantium
H0758 Cheng Pi橙皮 Bitter orangeCitrus aurantium
H1127 Guang Shan Zha广山楂 Chinese hawthornCrataegus pinnatifida
H0015 Ji Xing Zi急性子 Garden balsam seedImpatiens balsamina
H1201 Hu Er Cao虎耳草 Creeping rockfoilSaxifraga stolonifera
H0016 Ji Xue Cao积雪草 Asiatic pennywortCentella asiatica
H0421 Shan Zha Qing Gao山楂清膏 Chinese hawthornCrataegus pinnatifida
H0139 Lian Qiao连翘 Weeping forsythiaForsythia suspensa
H0466 Cai Fu Zi菜菔子 Semen raphaniRaphanus sativus
H0240 Mi Gan Cao蜜甘草 Glycyrrhiza inflataGlycyrrhiza uralensis
H0301 Ou Hindu lotus large rhizomeNelumbo nucifera
H0927 Da Huang Jin Gao大黄浸膏 Medicinal rhubarbRheum officinale
H0956 Dang Gui Gan Jin Gao当归干浸膏 NAAngelica sinensis
H0613 Wu Yue Ai五月艾 ArtemisiaArtemisia princeps
H0704 Yan Guan Huang Bai盐关黄柏 Amur cork treePhellodendron amurense
H0314 Pu Gong Ying蒲公英 Mongolian dandelionTaraxacum mongolicum
H0154 Ai Ye You艾叶油 Argy wormwood leafArtemisia argyi
H0519 Suo Yang锁阳 Songaria cynomoriumCynomorium songaricum
H0104 Bai Zhu白术 Largehead atractylodesAtractylodes macrocephala
H0571 Tu Gan Cao土甘草 Glycyrrhiza inflataGlycyrrhiza uralensis
H1029 Fang Er Cha方儿茶 khair in hindiSenegalia catechu
H0273 Mu Tong木通 Fiveleaf akebiaAkebia quinata
H1075 Gan Cao Liu Jin Gao甘草流浸膏 Glycyrrhiza inflataGlycyrrhiza uralensis
H1222 Huai Hua槐花 flower bud of japanese pagodatreeSophora japonica
H0278 Nan Ban Lan Gen Jin Gao Fen南板蓝根浸膏粉 Indigowoad rootBaphicacanthus cusia
H0103 Ai Ye艾叶 Argy wormwood leafArtemisia argyi
H1072 Gan Cao Gao甘草膏 Glycyrrhiza inflataGlycyrrhiza uralensis
H1224 Huai Jiao槐角 pod of japanese pagodatreeSophora japonica
H1169 He Ye荷叶 Hindu lotus leafNelumbo nucifera
H0818 Zhi Zi栀子 Cape jasmine fruitGardenia jasminoides
H0419 Shan Zha山楂 Chinese hawthornCrataegus pinnatifida
H0141 Lian Zi Xin莲子心 Hindu lotus plumuleNelumbo nucifera
H1046 Feng Xian Tou Gu Cao凤仙透骨草 Spotted snapweedImpatiens balsamina
H0988 Ding Gong Teng丁公藤 Obtuseleaf Erycibe StemErycibe obtusifolia
H0614 Wu Zhao Long五爪龙 Cairo morninggloryIpomoea cairica
H0413 Shan Lang Dang山莨菪 NAAnisodus tanguticus
H0733 Ye Shan Zha野山楂 nippon bawthornCrataegus pinnatifida
H1244 Huang Miao黄苗 NATaraxacum mongolicum
H0820 Chong Lou重楼 Paris rootRhizoma paridis
H0372 San Bai Bang三百棒 Chinese asparagusAsparagus cochinchinensis
H0418 Shan Yin Chen山茵陈 Capillary wormwoodArtemisia capillaris
H1138 Bai Jiang Cao败酱草 All - grass of dahurian patriniaThlaspi arvense
H0612 Cao Shan Hu Jin Gao草珊瑚浸膏 NASarcandra glabra
H1066 Gan Cao甘草 Glycyrrhiza inflataGlycyrrhiza uralensis
H0269 Mu Gua木瓜 Chinese floweringquinceChaenomeles sinensis
H1016 Du Zhong Tan杜仲炭 EucommiaEucommia ulmoides
H1230 Huang Bai Fen黄柏粉 Amur corktreePhellodendron amurense
H1067 Gan Cao Fen甘草粉 Glycyrrhiza inflataGlycyrrhiza uralensis
H0277 Nan Ban Lan Gen南板蓝根 Indigowoad rootBaphicacanthus cusia
H0095 Gou Qi Zi枸杞子 Chinese wolfberry fruitLycium chinense
H0424 Shan Zhi山栀 Cape jasmineGardenia jasminoides
H0094 Gou Qi枸杞 Chinese wolfberry fruitLycium chinense
H0065 Jin Yin Hua Ti Qu Ye金银花提取液 Japanese honeysuckleLonicera japonica
H1004 Bai Cha白茶 White teaCamellia sinensis
H1017 Du Zhong Ye杜仲叶 Eucommia leafEucommia ulmoides
H1188 Hong Hua红花 SafflowerCarthamus tinctorius
H0304 Ou Pian藕片 Hindu lotus large rhizomeNelumbo nucifera
H0368 Rou Gui Zi肉桂子 CassiabarktreeCinnamomum cassia
H0958 Dang Shen党参 Pilose asiabellCodonopsis pilosula
H0302 Ou Fen藕粉 Hindu lotus large rhizomeNelumbo nucifera
H0928 Da Huang Liu Jin Gao大黄流浸膏 Medicinal rhubarbRheum officinale
H1045 Feng Xian Hua凤仙花 Spotted snapweedImpatiens balsamina
H0354 Ren Dong Teng忍冬藤 Japanese honeysuckle vineLonicera japonica
H0866 Chuan Bi Xie川萆薢 Sichuan castor seedDioscorea septemloba
H0064 Jin Yin Hua金银花 Japanese honeysuckleLonicera japonica
H0396 Sang Ye桑叶 White mulberry leafMorus alba
H1000 Dong Gua Zi冬瓜子 Chinese waxgourd seedBenincasa hispida
H0536 Tian Di Ding甜地丁 Manyflower gueldenstaedtid herbViola philippica
H0391 Sang Pi桑皮 Prepared root-bark white mulberryMorus alba
H1074 Gan Cao Jin Gao甘草浸膏 Glycyrrhiza inflataGlycyrrhiza uralensis
H0397 Sang Zhi桑枝 White mulberry branchMorus alba
H0998 Dong Gua Pi冬瓜皮 Chinese waxgourd peelBenincasa hispida
H1070 Gan Cao Gan Gao Fen甘草干膏粉 Glycyrrhiza inflataGlycyrrhiza uralensis
H0705 Yan Hu Lu Ba盐胡芦巴 FenugreekTrigonella foenum-graecum
H1220 Hua Xiang Shu Guo化香树果 NAPlatycarya strobilacea
H0422 Shan Zha Tan山楂炭 Chinese hawthornCrataegus pinnatifida
H1225 Huai Mi槐米 NASophora japonica
H0420 Shan Zha Chou Gao山楂稠膏 Chinese hawthornCrataegus pinnatifida
H0053 Jin Lian Hua金莲花 Chinese globeflowerTrollius chinensis
H0472 Shu Da Huang熟大黄 NARheum palmatum
H0626 Xi Nan Huang Qin西南黄芩 Yunnan skullcapScutellaria amoena
H1069 Gan Cao Gan Gao甘草干膏 Glycyrrhiza inflataGlycyrrhiza uralensis
H0125 Lai Fu莱菔 Garden radishRaphanus sativus
H0932 Ba Qia菝葜 Chinaroot greenbrierSmilax china
H0570 Tu Fu Ling土茯苓 Glabrous greenbrierSmilax glabra
H0366 Rou Gui肉桂 CassiabarktreeCinnamomum cassia
H0540 Tian Ji Huang田基黄 all - grass of japanese st. johnswortGrangea maderaspatana
H0847 Zi He Che紫河车 Human placentaHomo sapiens
H0428 Shang Lu商陆 Indian pokeweedPhytolacca esculenta
H1231 Huang Bai Tan黄柏炭 Amur corktreePhellodendron amurense
H0140 Lian Zi莲子 Hindu lotus seedNelumbo nucifera
H1228 Huang Bai黄柏 Amur corktreePhellodendron amurense
H1071 Gan Cao Gan Jin Gao甘草干浸膏 Glycyrrhiza inflataGlycyrrhiza uralensis
H1221 Hua Xiang Shu Guo Xu化香树果序 NAPlatycarya strobilacea
H0335 Qin Pi秦皮 bark of largeleaf chinese ashCortex fraxini
H0585 Tu Yin Chen Hao土茵陈蒿 Capillary wormwoodArtemisia capillaris
H0325 Qian Jin Zi千金子 Caper euphorbia seedEuphorbia lathyris
H0537 Tian Dong天冬 Cochinchinese asparagus rootAsparagus cochinchinensis
H1115 Guan Huang Bai关黄柏 Amur cork treePhellodendron amurense
H0035 Bai Su Zi白苏子 Common perilla fruitPerilla frutescens
H1139 Gui Zhi桂枝 Cassiabarktree twigCinnamomum cassia
H0083 Jiu Jie Cha九节茶 Glabrous sarcandraSarcandra glabra
H0746 Yin Chen Hao Gan Jin Gao茵陈蒿干浸膏 Capillary wormwoodArtemisia capillaris
H0528 Tao Jin Niang Gen桃金娘根 Downy rosemyrtle rootRhodomyrtus tomentosa
H0640 Xiang Fu香附 Nutgrass galingaleCyperus rotundus
H0813 Zhi Shi枳实 Seville orange young fruitCitrus aurantium
H0444 Sheng Gan Cao生甘草 Glycyrrhiza inflataGlycyrrhiza uralensis