Target Description

Type Detail
Target ID T53KY7
Protein Name Cystic fibrosis transmembrane conductance regulator
Uniprot ID P13569
Protein Name Alias CFTR;  ATP-binding cassette sub-family C member 7;  Channel conductance-controlling ATPase;  EC 5.6.1.6;  cAMP-dependent chloride channel
Gene ID 1080
Gene Symbol CFTR
Gene Alias ABCC7
TTD T55654: Successful target
Pfam PF00664 ; PF00005 ; PF14396
GO
0016887:ATPase activity

0055085:transmembrane transport

0005634:nucleus

0006695:cholesterol biosynthetic process

0055038:recycling endosome membrane

0005829:cytosol

0005765:lysosomal membrane

0051087:chaperone binding

0016020:membrane

0032991:protein-containing complex

0015108:chloride transmembrane transporter activity

0016853:isomerase activity

0045921:positive regulation of exocytosis

1902476:chloride transmembrane transport

0016579:protein deubiquitination

0034976:response to endoplasmic reticulum stress

0005254:chloride channel activity

1902161:positive regulation of cyclic nucleotide-gated ion channel activity

0030660:Golgi-associated vesicle membrane

0019899:enzyme binding

0050891:multicellular organismal water homeostasis

1904322:cellular response to forskolin

0015106:bicarbonate transmembrane transporter activity

0034707:chloride channel complex

0005789:endoplasmic reticulum membrane

0030165:PDZ domain binding

0009986:cell surface

0051454:intracellular pH elevation

0048240:sperm capacitation

0042626:ATPase-coupled transmembrane transporter activity

0016021:integral component of membrane

0005524:ATP binding

0035377:transepithelial water transport

0005260:intracellularly ATP-gated chloride channel activity

0030301:cholesterol transport

0035774:positive regulation of insulin secretion involved in cellular response to glucose stimulus

0010008:endosome membrane

0055037:recycling endosome

0035973:aggrephagy

0015701:bicarbonate transport

0060081:membrane hyperpolarization

1902943:positive regulation of voltage-gated chloride channel activity

0030669:clathrin-coated endocytic vesicle membrane

0005886:plasma membrane

0016324:apical plasma membrane

0005769:early endosome

0019869:chloride channel inhibitor activity

0005887:integral component of plasma membrane

0071320:cellular response to cAMP

0005737:cytoplasm

0061024:membrane organization

0106138:Sec61 translocon complex binding

0006904:vesicle docking involved in exocytosis

0031901:early endosome membrane

PDB 5TFI ; 5TF8 ; 6O2P ; 5UAK ; 5D3E ; 2BBT ; 6MSM ; 6UK1 ; 6GK4 ; 2PZG ; 5TFG ; 5TFJ ; 6GJS ; 5D2D ; 5TFB ; 1XMI ; 2BBO ; 3ISW ; 1XMJ ; 4WZ6 ; 2LOB ; 5TFF ; 5D3F ; 2PZF ; 6GKD ; 2PZE ; 5TFA ; 5TFC ; 5TFD ; 5TF7 ; 6GJQ ; 1NBD ; 3GD7 ; 6O1V ; 6HEP ; 6GJU ; 5TGK ; 2BBS
Drugbank DB06266 ; DB15444 ; DB04941 ; DB00171 ; DB01050 ; DB04395 ; DB11712 ; DB00887 ; DB02587 ; DB08820 ; DB09280 ; DB04522 ; DB01016 ; DB09213
KEGG hsa:1080

Related Compounds  (Total: 5)

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C0101
Name: Genistein
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C0242
Name: Naringenin
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C0243
Name: Naringin
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C0409
Name: S-Nitrosoglutathione
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C0627
Name: Matrine


Related Herbs  (Total: 113)

Herb idChinese Pin YinChinese CharacterEnglish NameLatin Name
H0088 Ju He橘核 Tangerine seedCitrus reticulata
H1227 Huai Zhi槐枝 NASophora japonica
H0111 Ku Shen苦参 Lightyellow sophoraSophora flavescens
H0651 Xiang Yuan香橼 Wilson citronCitrus medica
H1174 Hei Da Dou黑大豆 Black soyabeanGlycine max
H0926 Da Huang大黄 Medicinal rhubarbRheum officinale
H0360 Ren Zhong Bai人中白 Human urine sedimentHomo sapiens
H1217 Bai Mei Hua白梅花 Japanese apricot flowerPrunus mume
H1034 Fei Yang Cao飞杨草 NAEuphorbia hirta
H0950 Dan Shen Gan Jin Gao丹参干浸膏 The root of red-rooted salviaSalvia miltiorrhiza
H0152 Ling Zhi Jin Gao灵芝浸膏 NAGanoderma lucidum
H1124 Guang Jin Qian Cao广金钱草 Snowbellleaf tickcloverDesmodium styracifolium
H0644 Xiang Mao香茅 LemongrassCymbopogon citratus
H1133 Gui Jian Yu鬼箭羽 Winged euonymusEuonymus alatus
H1094 Ge Gen葛根 Lobed kudzuvine rootPueraria lobata
H1080 Gan Ge干葛 Lobed kudzuvine rootPueraria lobata
H0153 Ling Zhi(1)灵芝 Lucid ganodermaGanoderma lucidum
H0130 Lei Gong Teng雷公藤 Common threewingnutTripterygium wilfordii
H0667 Xiao Qing Pi小青皮 Green tangerine peelPericarpium citri reticulatae viride
H0802 Zhi Geng枳梗 NACitrus aurantium
H1240 Huang Jing Zi黄荆子 NAVitex negundo
H0804 Zhi Ke枳壳 Seville ora nge unripe fruitCitrus aurantium
H1073 Gan Cao Jie甘草节 Glycyrrhiza uralensis fischGlycyrrhiza uralensis
H0805 Zhi Ke Gan Jin Gao枳壳干浸膏 Seville ora nge unripe fruitCitrus aurantium
H0758 Cheng Pi橙皮 Bitter orangeCitrus aurantium
H0663 Xiao Ji小蓟 Setose thistleCirsium setosum
H0965 Deng Zhan Xi Xin灯盏细辛 Shortscape fleabaneErigeron breviscapus
H0240 Mi Gan Cao蜜甘草 Glycyrrhiza inflataGlycyrrhiza uralensis
H1007 Dou You豆油 Soybean oilGlycine max
H0084 Jiu Li Xiang九里香 Common jasminorangeMurraya paniculata
H0927 Da Huang Jin Gao大黄浸膏 Medicinal rhubarbRheum officinale
H0195 Ma Chi Xian马齿苋 PurslanePortulaca oleracea
H0574 Cao Dou Kou草豆蔻 Katsumada galangalAlpinia katsumadai
H1102 Gu Sui Bu骨碎补 Fortune’s drynaria rhizomeDrynaria fortunei
H0571 Tu Gan Cao土甘草 Glycyrrhiza inflataGlycyrrhiza uralensis
H1140 Guo Gang Long过岗龙 NAEntada phaseoloides
H1222 Huai Hua槐花 flower bud of japanese pagodatreeSophora japonica
H1075 Gan Cao Liu Jin Gao甘草流浸膏 Glycyrrhiza inflataGlycyrrhiza uralensis
H0278 Nan Ban Lan Gen Jin Gao Fen南板蓝根浸膏粉 Indigowoad rootBaphicacanthus cusia
H1072 Gan Cao Gao甘草膏 Glycyrrhiza inflataGlycyrrhiza uralensis
H1224 Huai Jiao槐角 pod of japanese pagodatreeSophora japonica
H1095 Ge Gen Gan Jin Gao葛根干浸膏 Lobed kudzuvine rootPueraria lobata
H0347 Qing Pi青皮 Green tangerine peelPericarpium citri reticulatae viride
H0792 Zhang Yu章鱼 Common atlantic octopusOctopus vulgaris
H0979 Di Yu地榆 Garden burnetSanguisorba officinalis
H0089 Ju Hong橘红 NACitri exocarpium rubrum
H0405 Shan Dou Gen山豆根 Tonkin sophora rootSophora subprostrata
H0129 Le Xian Cai勒苋菜 NAAmaranthus spinosus
H0166 Long Kui龙葵 Black nightshadeSolanum nigrum
H0046 Jin Gan金柑 Japanese kumquatFortunella japonica
H1066 Gan Cao甘草 Glycyrrhiza inflataGlycyrrhiza uralensis
H0031 Jiang Tan姜炭 Soybean pasteGlycine max
H0629 Xi Xin细辛 Siebold wildgingerAsarum sieboldii
H1067 Gan Cao Fen甘草粉 Glycyrrhiza inflataGlycyrrhiza uralensis
H0277 Nan Ban Lan Gen南板蓝根 Indigowoad rootBaphicacanthus cusia
H0026 Jiang Soybean pasteGlycine max
H0951 Dan Shen Jin Gao丹参浸膏 The root of red-rooted salviaSalvia miltiorrhiza
H0533 Teng Ku Shen藤苦参 NASophora flavescens
H0604 Wu Wei Teng五味藤 NASecuridaca inappendiculata
H0092 Ju Hua菊花 Florists chrysanthemum flowerChrysanthemum morifolium
H0602 Wu Mei Rou乌梅肉 EbonyPrunus mume
H0052 Jin Ju金橘 Oval kumquatFortunella margarita
H0582 Cao Dou Kou Ren草豆蔻仁 Katsumada galangalAlpinia katsumadai
H0995 Dong Chong Xia Cao冬虫夏草 AwetoCordyceps sinensis
H1247 Huang Qi黄芪 Membranous milkvetchAstragalus membranaceus
H0976 Di Qing Pi地青皮 NAPericarpium citri reticulatae viride
H0002 Hui Xiang茴香 Fennel fruitFoeniculum vulgare
H0852 Zi Tan紫檀 Burmacoast padaukPterocarpus indicus
H0928 Da Huang Liu Jin Gao大黄流浸膏 Medicinal rhubarbRheum officinale
H0719 Chen Pi陈皮 Dried tangerine peelPericarpium citri reticulatae
H0952 Dan Xiang Chi淡香豉 NAGlycine max
H0396 Sang Ye桑叶 White mulberry leafMorus alba
H0093 Ju Pi橘皮 Tangerine pericarpCitrus reticulata
H0391 Sang Pi桑皮 Prepared root-bark white mulberryMorus alba
H1161 Hang Ju杭菊 Chrysanthemum flowerChrysanthemum morifolium
H1074 Gan Cao Jin Gao甘草浸膏 Glycyrrhiza inflataGlycyrrhiza uralensis
H0164 Ban Zhi Lian半枝莲 Barbed skullcapScutellaria barbata
H0397 Sang Zhi桑枝 White mulberry branchMorus alba
H1070 Gan Cao Gan Gao Fen甘草干膏粉 Glycyrrhiza inflataGlycyrrhiza uralensis
H0446 Sheng Jiang生姜 Fresh common gingerZingiber officinale
H0601 Wu Mei乌梅 Japanese apricotPrunus mume
H0705 Yan Hu Lu Ba盐胡芦巴 FenugreekTrigonella foenum-graecum
H0980 Di Yu Tan地榆炭 Garden burnetSanguisorba officinalis
H0219 Man Shan Hong满山红 Dahurian rhododendronRhododendron dauricum
H0575 Tu Ku Shen土苦参 all-grass of hooker wingheadSophora flavescens
H0369 Bian Fu Ge蝙蝠葛 Asiatic moonseedMenispermum dauricum
H1215 Hua Ju Hong化橘红 Pummelo peelExocarpium citri grandis
H0652 Xiang Yuan Pi香橼皮 Wilson citronCitrus medica
H1225 Huai Mi槐米 NASophora japonica
H1098 Gou Ji狗脊 Cochinchina cudraniaCudrania cochinchinensis
H1250 Huang Qi Ti Qu Ye黄芪提取液 Membranous milkvetchAstragalus membranaceus
H0053 Jin Lian Hua金莲花 Chinese globeflowerTrollius chinensis
H0472 Shu Da Huang熟大黄 NARheum palmatum
H1096 Ge Hua葛花 flower bud of lobed kudzuvinePueraria lobata
H0027 Jiang Gao姜膏 Soybean pasteGlycine max
H1069 Gan Cao Gan Gao甘草干膏 Glycyrrhiza inflataGlycyrrhiza uralensis
H0932 Ba Qia菝葜 Chinaroot greenbrierSmilax china
H0570 Tu Fu Ling土茯苓 Glabrous greenbrierSmilax glabra
H0847 Zi He Che紫河车 Human placentaHomo sapiens
H1141 Guo Gang Long Jin Gao过岗龙浸膏 NAEntada phaseoloides
H0091 Ju Hong Pi橘红皮 Red tangerine peelExocarpium citri rubrum
H1071 Gan Cao Gan Jin Gao甘草干浸膏 Glycyrrhiza inflataGlycyrrhiza uralensis
H0949 Dan Shen丹参 The root of red-rooted salviaSalvia miltiorrhiza
H0457 Shi Er石耳 Rock-EarsUmbilicaria esculenta
H0192 Lv Yi Zhi Shi绿衣枳实 NAPoncirus trifoliata
H0467 Shi Shang Bai石上柏 Doederlein's spikemoss herbHerba selaginellae doederleinii
H0324 Qian Jin Ba千斤拔 root of philippine flemingiaRadix moghaniae philippinensis
H0906 Ci Wan刺苋 spiny amaranthAmaranthus spinosus
H1249 Huang Qi Jin Gao黄芪浸膏 Membranous milkvetchAstragalus membranaceus
H1248 Huang Qi Gan Jin Gao黄芪干浸膏 Membranous milkvetchAstragalus membranaceus
H0944 Dan Dou Gu淡豆鼓 NAGlycine max
H0813 Zhi Shi枳实 Seville orange young fruitCitrus aurantium
H0444 Sheng Gan Cao生甘草 Glycyrrhiza inflataGlycyrrhiza uralensis